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Opioid Receptor


Opioid receptors are a group of inhibitory G protein-coupled receptors with opioids as ligands.[1][2][3] The endogenous opioids are dynorphins, enkephalins, endorphins, endomorphins and nociceptin. The opioid receptors are ~40% identical to somatostatin receptors (SSTRs). Opioid receptors are distributed widely in the brain, and are found in the spinal cord and digestive tract.The endogenous opioid system is thought to be important in mediating complex social behaviors involved in the formation of stable, emotionally committed relationships.
  • Morphine hydrochloride EI1754

    Morphine hydrochloride是Narcotic opioid analgesic。

    More
  • ML 190 EI1709

    ML 190是选择性 κ opioid 受体拮抗剂。

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  • Naltrexone HCl EY1576

    Naltrexone Hydrochloride (盐酸纳曲酮) 是阿片受体拮抗剂。

    More
  • Naloxone HCl EY1177

    Naloxone盐酸盐是阿片类拮抗剂,对阿片受体的IC50为3 nM。

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  • (+)-Matrine EY1462

    Matrine是来源于植物的生物碱,有抗肿瘤活性,是kappa阿片受体激动剂。

    More
  • Morphine hydrochloride EI1754

    Morphine hydrochloride是Narcotic opioid analgesic。

    More
  • ML 190 EI1709

    ML 190是选择性 κ opioid 受体拮抗剂。

    More
  • Naltrexone HCl EY1576

    Naltrexone Hydrochloride (盐酸纳曲酮) 是阿片受体拮抗剂。

    More
  • Naloxone HCl EY1177

    Naloxone盐酸盐是阿片类拮抗剂,对阿片受体的IC50为3 nM。

    More
  • (+)-Matrine EY1462

    Matrine是来源于植物的生物碱,有抗肿瘤活性,是kappa阿片受体激动剂。

    More
  • Morphine hydrochloride EI1754

    Morphine hydrochloride是Narcotic opioid analgesic。

    More
  • ML 190 EI1709

    ML 190是选择性 κ opioid 受体拮抗剂。

    More
  • Naltrexone HCl EY1576

    Naltrexone Hydrochloride (盐酸纳曲酮) 是阿片受体拮抗剂。

    More
  • Naloxone HCl EY1177

    Naloxone盐酸盐是阿片类拮抗剂,对阿片受体的IC50为3 nM。

    More
  • (+)-Matrine EY1462

    Matrine是来源于植物的生物碱,有抗肿瘤活性,是kappa阿片受体激动剂。

    More
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